SCHEMBL9215978

SCHEMBL9215978

O=C1Cc2cc3c(cc2CCN1CC1CCN(CCCc2cccnc2)C1)OCO3

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.39
PDE6D O43924 1/20 0.39
PDE6A P16499 1/20 0.39
PDE6G P18545 1/20 0.39
PDE6B P35913 1/20 0.39
PDE6C P51160 1/20 0.39
PDE6H Q13956 1/20 0.39
PDE11A Q9HCR9 1/20 0.39
CYP19A1 P11511 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
NAMPT P43490 1/20 0.35
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216543 0.95 LTA4H (0.39) PDE5APDE6DPDE6APDE6GPDE6B
Hydrochloric Acid SCHEMBL9739565 0.94 LTA4H (0.38) PDE5APDE6DPDE6APDE6GPDE6B
SCHEMBL9206838 0.90 ACHE (0.35) CYP19A1CYP11B1CYP11B2ACHE
Hydrochloric Acid SCHEMBL9213791 0.89 ACHE (0.37) PDE5APDE6DPDE6APDE6GPDE6B
Hydrochloric Acid SCHEMBL9741715 0.88 ACHE (0.34) ACHE
SCHEMBL9212426 0.86 PDE6D (0.39) PDE5APDE6DPDE6APDE6GPDE6B
SCHEMBL9213603 0.85 GRM5 (0.38) PDE5APDE6DPDE6APDE6GPDE6B
Hydrochloric Acid SCHEMBL9215725 0.85 GRM5 (0.38) PDE5APDE6DPDE6APDE6GPDE6B
SCHEMBL9213488 0.84 NAMPT (0.39) CYP19A1CYP11B1CYP11B2NAMPT
Hydrochloric Acid SCHEMBL9740467 0.83 NAMPT (0.38) CYP19A1CYP11B1CYP11B2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed