SCHEMBL9210936

SCHEMBL9210936

CCCCn1nnc(-c2cnc3ccccn3c2=O)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.40
NPC1 O15118 7/20 0.39
RAB9A P51151 7/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 6/20 0.38
ALDH1A1 P00352 5/20 0.38
TP53 P04637 3/20 0.38
HPGD P15428 3/20 0.38
DDX3X O00571 1/20 0.38
USP2 O75604 2/20 0.37
TSHR P16473 2/20 0.36
KDM4E B2RXH2 2/20 0.36
HSD17B10 Q99714 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
HTT P42858 1/20 0.36
GSK3B P49841 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217990 0.93 NPC1 (0.39) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL9217238 0.88 SMN1; SMN2 (0.40) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL9253405 0.85 NPC1 (0.37) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL9218231 0.83 NPC1 (0.38) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL9210165 0.82 ALDH1A1 (0.43) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL9212327 0.81 ADORA3 (0.38) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL9262200 0.80 MAPT (0.50) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL9260875 0.79 ESR1 (0.47) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL9259873 0.78 TRPV1 (0.38)
SCHEMBL9211054 0.78 LMNA (0.44) MAPTNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5475000-A Antiulcer agents CHINOIN GYOGYSZER-ES VEGYESZETI TERMEKEK GYARA RT. (HU) 1995-12-12 US disclosed
EP-0641340-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO- 1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN Gyogyszer és Vegyészeti Termékek Gyára RT. (HU) 1995-03-08 EP disclosed
WO-1993004065-A1 NEW 3-(SUBSTITUTED TETRAZOLYL)-4-OXO-4H-PYRIDO-[1,2-a]PYRIMIDINES, SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESS FOR PREPARING SAME CHINOIN GYÓGYSZER- ÉS VEGYÉSZETI TERMÉKEK GYÁRA RT. (HU) 1993-03-04 WO disclosed