SCHEMBL9218155

SCHEMBL9218155

CCOC(=O)[C@H](CO)NC(=O)[C@H](CC(=O)OCc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 1/20 0.53
KLK5 Q9Y337 1/20 0.53
CTSS P25774 4/20 0.48
MMP9 P14780 1/20 0.48
PPARA Q07869 2/20 0.47
SYK P43405 1/20 0.47
CTSK P43235 2/20 0.47
REN P00797 3/20 0.47
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CACNA1B Q00975 4/20 0.46
PSMB5 P28074 1/20 0.46
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
PPARG P37231 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9217713 0.94 REN (0.50) KLK7KLK5CTSSMMP9SYK
SCHEMBL27510152 0.92 CTSS (0.53) KLK7KLK5CTSSMMP9SYK
SCHEMBL9217707 0.89 SYK (0.46) KLK7KLK5CTSSMMP9SYK
SCHEMBL8430460 0.89 KLK7 (0.54) KLK7KLK5CTSSMMP9PPARA
SCHEMBL12292883 0.87 PPARA (0.55) KLK7KLK5CTSSPPARASYK
SCHEMBL7294995 0.86 CTSS (0.56) KLK7KLK5CTSSMMP9PPARA
SCHEMBL14037329 0.86 SYK (0.53) KLK7KLK5CTSSSYKCTSK
SCHEMBL25491606 0.86 KLK7 (0.59) KLK7KLK5CTSSPPARASYK
SCHEMBL5419241 0.86 KLK7 (0.59) KLK7KLK5CTSSPPARASYK
SCHEMBL12292731 0.85 BACE1 (0.51) CTSSPPARACTSKRENCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed