SCHEMBL9218176

SCHEMBL9218176

O=Cc1cc(Br)c(OCCCCCCc2ccccc2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 1/20 0.47
THRA P10827 4/20 0.43
THRB P10828 4/20 0.43
S1PR1 P21453 3/20 0.40
S1PR3 Q99500 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
FFAR1 O14842 1/20 0.40
S1PR5 Q9H228 1/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7163250 1.00 ALDH1A1 (0.47) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL7164257 0.99 ALDH1A1 (0.48) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL7161998 0.94 LMNA (0.49) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL7168103 0.90 ALDH1A1 (0.50) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL1981552 0.83 HPGD (0.52) ALDH1A1LMNAMAPTS1PR1S1PR3
SCHEMBL14195850 0.81 ALDH1A1 (0.55) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL3955227 0.80 THRA (0.57) ALDH1A1LMNAMAPTTHRATHRB
SCHEMBL9218172 0.80 FFAR1 (0.43) ALDH1A1LMNATHRATHRBS1PR1
SCHEMBL7163248 0.80 FFAR1 (0.43) ALDH1A1LMNATHRATHRBS1PR1
SCHEMBL8408121 0.79 THRA (0.49) THRATHRBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed
EP-0269859-A2 Pyrazolotriazine compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-06-08 EP disclosed