Morphine

Morphine

SCHEMBL9219855

CN1CC[C@]23c4c5ccc(O)c4O[C@H]2[C@@H](O)C=C[C@H]3[C@H]1C5.O=C(O)[C@H]1O[C@H](O)[C@H](O)[C@@H](O)[C@@H]1O

nearest known ligand 0.75

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

OPRM1

The experimentally established mechanism targets of Morphine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
OPRM1 known ✓ P35372 7/20 0.75
OPRD1 P41143 7/20 0.75
OPRK1 P41145 5/20 0.75
MRGPRX2 Q96LB1 3/20 0.75
SLC22A1 O15245 1/20 0.75
ADRA2A P08913 1/20 0.75
ARRB1 P49407 1/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Morphine SCHEMBL8374708 0.88 OPRD1 (0.90) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL15055206 0.88 OPRD1 (0.90) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL149700 0.88 OPRD1 (0.90) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL2443249 0.87 OPRD1 (0.89) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL27547724 0.87 OPRD1 (0.96) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL24599520 0.87 OPRD1 (1.00) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL2997 0.87 OPRD1 (1.00) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL8049464 0.87 OPRD1 (1.00) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL5183254 0.87 OPRD1 (1.00) OPRM1OPRD1OPRK1MRGPRX2SLC22A1
Morphine SCHEMBL13076870 0.87 OPRD1 (1.00) OPRM1OPRD1OPRK1MRGPRX2SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995005831-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING MORPHINE-6-GLUCURONIDE FOR THE TREATMENT OF PAIN EURO-CELTIQUE S.A. (LU) 1995-03-02 WO disclosed