SCHEMBL9224600

SCHEMBL9224600

C1CCN(c2nc(N3CCCC3)nc(N3CC[N]CC3)n2)C1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.56
SMN1; SMN2 Q16637 2/20 0.54
USP2 O75604 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
MAPK1 P28482 4/20 0.52
ALDH1A1 P00352 3/20 0.52
NPC1 O15118 1/20 0.52
GALR3 O60755 1/20 0.52
TP53 P04637 1/20 0.52
RAB9A P51151 1/20 0.52
MEN1 O00255 5/20 0.50
KMT2A Q03164 5/20 0.50
HTT P42858 1/20 0.50
RECQL P46063 1/20 0.50
ATM Q13315 1/20 0.50
LMNA P02545 3/20 0.47
CYP2C9 P11712 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1975340 0.86 HRH1 (0.70) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL11208162 0.83 SMN1; SMN2 (0.71) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL9722891 0.83 CASP1 (0.67) HRH1SMN1; SMN2USP2TDP1KMT2A
SCHEMBL9730702 0.80 SMN1; SMN2 (0.68) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL9803306 0.80 HRH1 (0.62) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL9073359 0.74 HRH1 (0.56) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL29274357 0.74 HRH1 (0.56) HRH1SMN1; SMN2USP2TDP1MAPK1
Triethylenemelamine SCHEMBL8359 0.73 HRH1 (0.52) HRH1SMN1; SMN2USP2TDP1MAPK1
SCHEMBL10494023 0.72 SMN1; SMN2 (0.58) HRH1SMN1; SMN2USP2TDP1MAPK1
Hydrochloric Acid SCHEMBL31046022 0.72 HRH1 (0.54) HRH1SMN1; SMN2USP2TDP1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380840-A Treating spinal trauma, head injury, subarachnoid hemorrhage; reduced side effects THE UPJOHN COMPANY (US) 1995-01-10 US claimed
EP-0354920-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1990-02-21 EP claimed
WO-1988007527-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1988-10-06 WO claimed
EP-0238545-A1 C 20? THROUGH C 26? AMINO STEROIDS. UPJOHN CO (US) 1987-09-30 EP claimed
WO-1987001706-A2 C20 THROUGH C26 AMINO STEROIDS THE UPJOHN COMPANY (US) 1987-03-26 WO claimed
US-4996318-A Amino-9,10-secosteroids useful for treating head injury, spinal cord trauma or stroke THE UPJOHN COMPANY (US) 1991-02-26 US disclosed
EP-0354920-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1990-02-21 EP disclosed
WO-1988007527-A1 AMINO-9,10-SECOSTEROIDS THE UPJOHN COMPANY (US) 1988-10-06 WO disclosed