SCHEMBL9224607

SCHEMBL9224607

OB(O)c1ccnc(-c2cc(B(O)O)ccn2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.42
CCR5 P51681 2/20 0.42
CCR8 P51685 2/20 0.42
ENPP2 Q13822 7/20 0.39
PLG P00747 1/20 0.39
F12 P00748 1/20 0.39
F11 P03951 1/20 0.39
KLKB1 P03952 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
PRSS3 P35030 1/20 0.39
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MGLL Q99685 1/20 0.37
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30151430 1.00 CCR1 (0.42) CCR1CCR5CCR8ENPP2PLG
SCHEMBL3873666 0.88 KDM4E (0.54) CCR1CCR5CCR8CA1CA2
SCHEMBL29955214 0.83 ASIC3 (0.53) ENPP2PLGF12F11KLKB1
SCHEMBL21527865 0.83 ASIC3 (0.53) ENPP2PLGF12F11KLKB1
SCHEMBL24610115 0.83 PLG (0.33) CCR1CCR5CCR8ENPP2PLG
SCHEMBL25224336 0.82 JMJD6 (0.56) CCR1CCR5CCR8KDM4E
SCHEMBL31333872 0.80 NPC1 (0.44) PLGF12F11KLKB1PRSS1
SCHEMBL15332828 0.80 NPC1 (0.44) PLGF12F11KLKB1PRSS1
SCHEMBL29950674 0.79 IDO1 (0.46) PLGF12F11KLKB1PRSS1
SCHEMBL29953273 0.79 ALDH1A1 (0.45) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7133283-A None JP disclosed
JP-H07133283-A AROMATIC BETA-DIMINE-BASED COMPOUND RES DEV CORP OF JAPAN 1995-05-23 JP disclosed