Declopramide

Declopramide

SCHEMBL922516

CCN(CC)CCNC(=O)c1ccc(N)c(Cl)c1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.66
ALDH1A1 P00352 4/20 0.66
SLC22A1 O15245 2/20 0.66
SLC22A2 O15244 1/20 0.66
TSHR P16473 1/20 0.66
ACHE P22303 1/20 0.66
MAPK1 P28482 1/20 0.66
CYP2C19 P33261 1/20 0.66
BLM P54132 2/20 0.64
PMP22 Q01453 1/20 0.64
KCNH2 Q12809 2/20 0.59
HTR3E A5X5Y0 1/20 0.59
HTR3B O95264 1/20 0.59
MPO P05164 1/20 0.59
CYP1A2 P05177 1/20 0.59
ADRA2A P08913 1/20 0.59
CYP2D6 P10635 1/20 0.59
DRD2 P14416 1/20 0.59
ADRA2C P18825 1/20 0.59
DRD4 P21917 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Declopramide SCHEMBL30719968 1.00 LMNA (0.66) LMNAALDH1A1SLC22A1SLC22A2TSHR
Declopramide SCHEMBL6436822 0.99 LMNA (0.67) LMNAALDH1A1SLC22A1SLC22A2TSHR
Declopramide SCHEMBL5925509 0.96 ALDH1A1 (0.61) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL18768840 0.87 HPGD (0.63) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL2956109 0.87 ALDH1A1 (0.71) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL3435195 0.86 LMNA (0.52) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL12886918 0.85 ALDH1A1 (0.68) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL5924476 0.85 ALDH1A1 (0.68) LMNAALDH1A1SLC22A1SLC22A2TSHR
SCHEMBL10079549 0.84 SMN1; SMN2 (0.56) LMNAALDH1A1TSHRCYP1A2CYP2D6
SCHEMBL3435778 0.82 SMN1; SMN2 (0.60) LMNAALDH1A1TSHRKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 298 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250259704-A1 SYSTEMS AND METHODS FOR CELL-FREE ITERATIVE SITE SATURATION MUTAGENESIS AND ITS APPLICATION FOR THE DIRECTED EVOLUTION OF ENZYMES CATALYZING UNNATURAL REACTIONS U.S. DEPARTMENT OF ENERGY 2025-08-14 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
WO-2023250524-A1 SYSTEMS AND METHODS FOR CELL-FREE ITERATIVE SITE SATURATION MUTAGENESIS AND ITS APPLICATION FOR THE DIRECTED EVOLUTION OF ENZYMES CATALYZING UNNATURAL REACTIONS NORTHWESTERN UNIVERSITY (US) 2023-12-28 WO claimed
EP-2459227-B1 Prodrugs containing an aromatic amine connected by an amide bond to a carrier ASCENDIS PHARMA AS (DK) 2021-03-17 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20120156260-A1 Prodrugs Containing an Aromatic Amine Connected By an Amido Bond to a Linker ASCENDIS PHARMA A/S (DK) 2012-06-21 US claimed
EP-2459227-A1 PRODRUGS CONTAINING AN AROMATIC AMINE CONNECTED BY AN AMIDO BOND TO A LINKER Ascendis Pharma A/S (DK) 2012-06-06 EP claimed
WO-2011012722-A1 PRODRUGS CONTAINING AN AROMATIC AMINE CONNECTED BY AN AMIDO BOND TO A LINKER ASCENDIS PHARMA AS (DK) 2011-02-03 WO claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
WO-2009045504-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER AND MODULATING SIGNAL TRANSDUCTION AND METABOLISM PATHWAYS PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2009-04-09 WO claimed
EP-1393277-A1 USE OF NFKB INHIBITORS TO TREAT DRY EYE DISORDERS Alcon, Inc. (CH) 2004-03-03 EP claimed
US-6696453-B2 ADMINISTERING NF- KAPPA B INHIBITORS FOR THERAPY OF DRY EYES ALCON, INC. (CH) 2004-02-24 US claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
WO-2002095704-A9 USE OF NF-KAPPA-B INHIBITORS TO TREAT DRY EYE DISORDERS ALCON INC (CH) 2003-02-27 WO claimed
US-20030008854-A1 Use of NF-kappabeta inhibitors to treat dry eye disorders ALCON, INC. 2003-01-09 US claimed
WO-2002095393-A2 DRUG EVOLUTION: DRUG DESIGN AT HOT SPOTS NATIONAL RESEARCH COUNCIL OF CANADA (CA) 2002-11-28 WO claimed
WO-2002095704-A1 USE OF NF-KAPPA-B INHIBITORS TO TREAT DRY EYE DISORDERS ALCON, INC. (CH) 2002-11-28 WO claimed
EP-0927030-A4 USE OF ARYL N-SUBSTITUTED CARBOXAMIDES TO KILL TUMORS OXIGENE INC (US) 2000-01-26 EP claimed
EP-0927030-A1 USE OF ARYL N-SUBSTITUTED CARBOXAMIDES TO KILL TUMORS OXIGENE, INC. (US) 1999-07-07 EP claimed
WO-1997032576-A1 USE OF ARYL N-SUBSTITUTED CARBOXAMIDES TO KILL TUMORS OXIGENE, INC. (US) 1997-09-12 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120156260-A1 Prodrugs Containing an Aromatic Amine Connected By an Amido Bond to a Linker DAO, DNPEP, DDC LMNA 759/4885ALDH1A1 899/4885SLC22A1 362/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.