SCHEMBL9225470

SCHEMBL9225470

C[C@@H](O)C(C(=O)OCc1ccccc1)N1C(=O)C(N2C(=O)c3ccccc3C2=O)C1CO

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 3/20 0.47
MAPK1 P28482 1/20 0.42
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
ELANE P08246 7/20 0.38
CTRB1 P17538 1/20 0.37
CDC25B P30305 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9225461 1.00 AVPR1A (0.47) AVPR1AMAPK1CYP3A4CYP2D6CYP2C9
SCHEMBL9224938 0.87 ACHE (0.43) AVPR1A
SCHEMBL9224944 0.87 ACHE (0.43) AVPR1A
SCHEMBL9219422 0.84 AVPR1A (0.35) AVPR1ACYP3A4CYP2C19HSD11B1
SCHEMBL9219312 0.84 AVPR1A (0.44) AVPR1AMAPK1CYP3A4CYP2D6CYP2C9
SCHEMBL9219306 0.84 AVPR1A (0.44) AVPR1AMAPK1CYP3A4CYP2D6CYP2C9
SCHEMBL9225933 0.83 AVPR1A (0.68) AVPR1AMAPK1CYP3A4CYP2D6CYP2C9
SCHEMBL9225930 0.83 AVPR1A (0.68) AVPR1AMAPK1CYP3A4CYP2D6CYP2C9
SCHEMBL9227516 0.81 HTR2A (0.37) AVPR1ARAB9AALDH1A1
SCHEMBL9228503 0.78 ALDH1A1 (0.42) MAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0282895-B1 2-oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMA CO LTD (JP) 1995-06-07 EP disclosed
US-5037976-A Antimicrobial Agent OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-08-06 US disclosed
US-4898859-A 2-Oxa-isocephem compounds and compositions containing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-02-06 US disclosed
EP-0282895-A2 2-oxa-isocephem compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-09-21 EP disclosed