SCHEMBL9229872

SCHEMBL9229872

CCOC(=O)C1(C(=O)N(CC)Cc2ccccc2)CC(=O)N(Cc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
LMNA P02545 3/20 0.41
TSHR P16473 3/20 0.41
MAPK1 P28482 2/20 0.41
NPC1 O15118 1/20 0.41
ALOX15 P16050 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TRPM8 Q7Z2W7 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
CASP3 P42574 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
TSPO P30536 2/20 0.39
OPRM1 P35372 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8881539 0.96 NPSR1 (0.41) ALDH1A1LMNATSHRMAPK1NPC1
SCHEMBL8881874 0.88 RAB9A (0.40) ALDH1A1LMNANPC1CASP3CYP3A4
SCHEMBL9233372 0.88 KDM4E (0.41) ALDH1A1LMNANPC1CASP3CYP3A4
SCHEMBL8881736 0.88 CASP3 (0.46) ALDH1A1LMNASLC6A4CASP3CYP3A4
SCHEMBL8882202 0.85 CASP3 (0.46) ALDH1A1LMNASLC6A4CASP3CYP3A4
SCHEMBL9231209 0.85 CYP3A4 (0.41) ALDH1A1LMNACASP3CYP3A4CYP2D6
SCHEMBL9232448 0.85 OPRM1 (0.47) ALDH1A1CASP3CYP3A4CYP2D6CYP2C9
SCHEMBL8881749 0.82 NPSR1 (0.43) LMNACYP2D6CYP2C9CYP2C19OPRM1
SCHEMBL8882513 0.80 CASP3 (0.47) ALDH1A1LMNACASP3CYP3A4CYP2D6
SCHEMBL9230909 0.78 CYP3A4 (0.46) ALDH1A1LMNASLC6A4CASP3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677522-A1 8-METHOXYQUINOLONECARBOXYLIC ACID DERIVATIVE YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-10-18 EP disclosed