SCHEMBL9230657

SCHEMBL9230657

N#CC1(NC(=O)c2ccccc2)CN(C(c2ccccc2)c2ccccc2)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 7/20 0.49
CTSK P43235 4/20 0.44
CTSB P07858 3/20 0.44
CTSS P25774 3/20 0.44
MAOB P27338 1/20 0.43
CYP3A4 P08684 5/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 2/20 0.42
USP2 O75604 3/20 0.41
HDAC1 Q13547 3/20 0.41
HDAC4 P56524 2/20 0.41
CYP1A2 P05177 1/20 0.41
KCNH2 Q12809 1/20 0.41
ALDH1A1 P00352 2/20 0.40
OPRD1 P41143 1/20 0.40
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
HIF1A Q16665 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19029710 0.78 CTSL (0.73) CTSLCTSKCTSBCTSSALDH1A1
SCHEMBL4841029 0.77 NPSR1 (0.45) CYP3A4CYP2D6CYP2C9CYP2C19USP2
SCHEMBL4837814 0.76 NPSR1 (0.44) CYP3A4CYP2D6CYP2C9CYP2C19USP2
SCHEMBL8055885 0.75 CTSL (0.74) CTSLCTSKCTSBCTSSALDH1A1
SCHEMBL5236409 0.73 NPSR1 (0.42) CYP3A4CYP2D6CYP2C9CYP2C19USP2
SCHEMBL1488545 0.72 NPSR1 (0.41) CTSLCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL29642581 0.71 CTSL (0.60) CTSLCTSKCTSBCTSS
SCHEMBL5527398 0.71 OPRL1 (0.49) CYP3A4CYP2D6CYP2C9USP2CYP1A2
SCHEMBL9233452 0.71 CTSL (0.56) CTSLCTSKCTSBCTSSALDH1A1
SCHEMBL9231743 0.71 OPRD1 (0.44) CTSLCTSKMAOBCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677522-A1 8-METHOXYQUINOLONECARBOXYLIC ACID DERIVATIVE YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-10-18 EP disclosed