SCHEMBL9232120

SCHEMBL9232120

CCCOC(=O)CC[N]Cc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.51
LMNA P02545 2/20 0.48
TOP2A P11388 2/20 0.45
ALDH1A1 P00352 4/20 0.44
ALOX5 P09917 1/20 0.40
LTA4H P09960 4/20 0.40
POLB P06746 2/20 0.40
APP P05067 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8852294 0.88 ALOX5 (0.48) TDP1TOP2AALDH1A1ALOX5LTA4H
SCHEMBL8852249 0.81 ALDH1A1 (0.51) TDP1LMNAALDH1A1LTA4HPOLB
SCHEMBL3851800 0.79 TDP1 (0.82) TDP1LMNAALDH1A1ALOX5APP
SCHEMBL8851560 0.79 ALOX5 (0.52) TDP1TOP2AALDH1A1ALOX5LTA4H
SCHEMBL13557789 0.78 TDP1 (0.68) TDP1LMNATOP2AALDH1A1ALOX5
SCHEMBL3954435 0.76 TDP1 (0.66) TDP1LMNATOP2AALOX5SMN1; SMN2
SCHEMBL650649 0.75 ALDH1A1 (0.63) TDP1LMNAALDH1A1ALOX5SMN1; SMN2
SCHEMBL10031001 0.75 ALDH1A1 (0.54) TDP1LMNATOP2AALDH1A1ALOX5
SCHEMBL16672928 0.75 TDP1 (0.54) TDP1LMNATOP2AALDH1A1POLB
SCHEMBL17578861 0.75 TDP1 (0.64) TDP1LMNATOP2AALOX5MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed