SCHEMBL9233255

SCHEMBL9233255

N#CC1(N(Cc2ccccc2)C(=O)c2ccccc2)CCN(Cc2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 5/20 0.52
CHRM3 P20309 5/20 0.52
OPRM1 P35372 2/20 0.49
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
ALDH1A1 P00352 2/20 0.45
CYP2D6 P10635 2/20 0.44
SIGMAR1 Q99720 1/20 0.44
ACHE P22303 2/20 0.44
KDM4E B2RXH2 1/20 0.43
OPRL1 P41146 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9228793 0.93 CHRM2 (0.47) CHRM2CHRM3OPRM1CTSSCTSK
SCHEMBL9234501 0.86 CHRM2 (0.46) CHRM2CHRM3CTSSCTSKALDH1A1
SCHEMBL9233113 0.84 CHRM2 (0.50) CHRM2CHRM3OPRM1ALDH1A1CYP2D6
SCHEMBL9232468 0.81 CHRM2 (0.53) CHRM2CHRM3OPRM1ALDH1A1ACHE
SCHEMBL9228402 0.80 ACHE (0.46) CHRM2CHRM3OPRM1CTSSCTSK
SCHEMBL2331319 0.79 OPRM1 (0.61) OPRM1ALDH1A1CYP2D6SIGMAR1ACHE
SCHEMBL5674633 0.78 OPRM1 (0.57) OPRM1ALDH1A1CYP2D6SIGMAR1OPRL1
SCHEMBL9232318 0.77 CYP3A4 (0.56) CHRM2CHRM3OPRM1ALDH1A1CYP2D6
SCHEMBL5671761 0.75 OPRM1 (0.53) OPRM1ALDH1A1CYP2D6SIGMAR1OPRL1
SCHEMBL9234493 0.74 CYP2D6 (0.48) CHRM2CHRM3ALDH1A1CYP2D6ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0677522-A1 8-METHOXYQUINOLONECARBOXYLIC ACID DERIVATIVE YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-10-18 EP disclosed