SCHEMBL923632

SCHEMBL923632

O=C(O)C1CCc2cccnc2C1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 6/20 0.44
FAAH O00519 4/20 0.43
KDM4E B2RXH2 1/20 0.41
CYP2C19 P33261 1/20 0.41
GRIN1 Q05586 4/20 0.40
GRIN2B Q13224 4/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17803288 0.89 IDH1 (0.50) IDH1FAAHKDM4ECYP2C19GRIN1
SCHEMBL3657715 0.87 DRD2 (0.47) IDH1FAAHKDM4ECYP2C19GRIN1
SCHEMBL3659200 0.87 DRD2 (0.47) IDH1FAAHKDM4ECYP2C19GRIN1
SCHEMBL3657710 0.87 DRD2 (0.47) IDH1FAAHKDM4ECYP2C19GRIN1
SCHEMBL5108390 0.85 KDM4E (0.41) IDH1FAAHKDM4ECYP2C19L3MBTL1
SCHEMBL369170 0.85 KDM4E (0.41) IDH1FAAHKDM4ECYP2C19L3MBTL1
Hydrochloric Acid SCHEMBL3241637 0.83 KDM4E (0.40) IDH1FAAHKDM4ECYP2C19L3MBTL1
SCHEMBL923515 0.82 FAAH (0.42) IDH1FAAHKDM4EGRIN1GRIN2B
SCHEMBL17803299 0.81 IDH1 (0.53) IDH1FAAHKDM4ECYP2C19L3MBTL1
Hydrochloric Acid SCHEMBL2883763 0.79 OPRL1 (0.45) IDH1FAAHKDM4ECYP2C19L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868020-B2 Quinolynylmethylimidizoles as therapeutic agents ALLERGAN, INC. (US) 2011-01-11 US disclosed
US-7868020-B2 Quinolynylmethylimidizoles as therapeutic agents ALLERGAN, INC. (US) 2011-01-11 US disclosed
US-7868020-B2 Quinolynylmethylimidizoles as therapeutic agents ALLERGAN, INC. (US) 2011-01-11 US disclosed
US-20100113516-A1 QUINOLYNYLMETHYLIMIDIZOLES AS THERAPEUTIC AGENTS ALLERGAN, INC. (US) 2010-05-06 US disclosed
US-20100113516-A1 QUINOLYNYLMETHYLIMIDIZOLES AS THERAPEUTIC AGENTS ALLERGAN, INC. (US) 2010-05-06 US disclosed
US-20100113516-A1 QUINOLYNYLMETHYLIMIDIZOLES AS THERAPEUTIC AGENTS ALLERGAN, INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113516-A1 QUINOLYNYLMETHYLIMIDIZOLES AS THERAPEUTIC AGENTS TUBB3, TUBB1, NQO2 IDH1 314/4885FAAH 3609/4885KDM4E 3836/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.