SCHEMBL9242577

SCHEMBL9242577

C=CCCNC(=O)CC(N)=O

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.38
TSHR P16473 4/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DDAH1 O94760 2/20 0.34
ECE1 P42892 1/20 0.33
FGFR4 P22455 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
LMNA P02545 1/20 0.31
ABCC4 O15439 1/20 0.30
MAPK1 P28482 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
ST14 Q9Y5Y6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6848895 0.80
SCHEMBL5804452 0.79
SCHEMBL14586442 0.79 MAPT (0.41) ALDH1A1TSHRMAPTSMN1; SMN2DDAH1
SCHEMBL28179346 0.77
SCHEMBL22856074 0.77 MAPT (0.46) ALDH1A1TSHRMAPTSMN1; SMN2LMNA
SCHEMBL4068835 0.77 SMN1; SMN2 (0.58) ALDH1A1TSHRMAPTSMN1; SMN2
SCHEMBL17884297 0.77 ALDH1A1 (0.46) ALDH1A1TSHRMAPTSMN1; SMN2DDAH1
SCHEMBL5466809 0.76
SCHEMBL28273001 0.76
SCHEMBL1344230 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0654025-A4 METHOD OF PREPARING OPTICALLY PURE PRECURSORS OF PAROXETINE. SEPRACOR INC (US) 1995-10-11 EP disclosed
EP-0654025-A1 METHOD OF PREPARING OPTICALLY PURE PRECURSORS OF PAROXETINE SEPRACOR, INC. (US) 1995-05-24 EP disclosed
WO-1994003428-A1 METHOD OF PREPARING OPTICALLY PURE PRECURSORS OF PAROXETINE SEPRACOR, INC. (US) 1994-02-17 WO disclosed
US-5258517-A Method of preparing optically pure precursors of paroxetine SEPRACOR, INC. (US) 1993-11-02 US disclosed