SCHEMBL9244337

SCHEMBL9244337

CC1(C)CCC(OCc2ccc3ccccc3n2)C(Cn2ccnc2)C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 7/20 0.35
ALOX5AP P20292 3/20 0.35
CALCA P06881 1/20 0.34
CYSLTR2 Q9NS75 1/20 0.34
CYSLTR1 Q9Y271 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
PGGT1B P53609 1/20 0.34
BRD4 O60885 1/20 0.33
CYP1A2 P05177 1/20 0.33
ALOX5 P09917 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9244356 1.00 PDE10A (0.35) PDE10AALOX5APCALCACYSLTR2CYSLTR1
SCHEMBL9241773 0.91 PDE10A (0.36) PDE10ACALCAFNTAFNTBPGGT1B
SCHEMBL9249928 0.84 REN (0.37) PDE10AALOX5APCYSLTR2CYSLTR1BRD4
SCHEMBL9249921 0.84 REN (0.37) PDE10AALOX5APCYSLTR2CYSLTR1BRD4
SCHEMBL9244520 0.82 POLB (0.47) FNTAFNTBPGGT1BCYP19A1
SCHEMBL9244542 0.82 POLB (0.47) FNTAFNTBPGGT1BCYP19A1
SCHEMBL9244600 0.81 CALCA (0.36) PDE10AALOX5APCALCACYSLTR2CYSLTR1
SCHEMBL9244604 0.81 CALCA (0.36) PDE10AALOX5APCALCACYSLTR2CYSLTR1
SCHEMBL8715873 0.81 CYSLTR1 (0.40) ALOX5APCYSLTR2CYSLTR1BRD4ALOX5
SCHEMBL9243625 0.81 CYSLTR1 (0.40) ALOX5APCYSLTR2CYSLTR1BRD4ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449785-A Fungicides with triazole groups HOFFMANN-LA ROCHE INC. (US) 1995-09-12 US disclosed
EP-0524439-A1 Novel cyclohexane and tetrahydropyran derivatives and antifungal compositions containing these derivatives F.HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT (CH) 1993-01-27 EP disclosed