SCHEMBL9245211

SCHEMBL9245211

C/C=C/CC1CCC(C#Cc2ccc(-c3ccc(Cl)c(F)c3)nc2)CC1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGES O14684 3/20 0.37
GRM2 Q14416 2/20 0.33
EGLN1 Q9GZT9 1/20 0.33
KMO O15229 1/20 0.32
CHRNB2 P17787 2/20 0.31
CHRNA2 Q15822 2/20 0.31
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
CHRNA4 P43681 1/20 0.31
BACE1 P56817 2/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
GRM5 P41594 1/20 0.30
MCHR1 Q99705 1/20 0.30
P2RX7 Q99572 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9246659 0.91 GRM2 (0.38) PTGESGRM2EGLN1CHRNB2CHRNA2
SCHEMBL9246397 0.88 CHRNB2 (0.32) PTGESEGLN1CHRNB2CHRNA2CHRNB4
SCHEMBL9245509 0.87 FFAR1 (0.33) MCHR1
SCHEMBL9250091 0.86 GRM5 (0.42) PTGESEGLN1CHRNB2CHRNA2CHRNB4
SCHEMBL9245099 0.86 MCHR1 (0.41) PTGESEGLN1CHRNB2CHRNA2CHRNB4
SCHEMBL9249257 0.85 PTGES (0.38) PTGESGRM2EGLN1KMOBACE1
SCHEMBL9249265 0.85 PTGES (0.38) PTGESGRM2EGLN1KMOBACE1
SCHEMBL9244989 0.85 PTGES (0.36) PTGESGRM2EGLN1KMOBACE1
SCHEMBL9244993 0.85 PTGES (0.36) PTGESGRM2EGLN1KMOBACE1
SCHEMBL9244982 0.85 PTGES (0.36) PTGESGRM2EGLN1KMOBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US disclosed