SCHEMBL9250091

SCHEMBL9250091

C/C=C/CC1CCC(C#Cc2ccc(-c3ccc(F)cc3)nc2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.42
EGLN1 Q9GZT9 1/20 0.34
PTGES O14684 2/20 0.33
CHRNB2 P17787 2/20 0.32
CHRNA2 Q15822 2/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
AURKA O14965 1/20 0.32
ABL1 P00519 1/20 0.32
NTRK1 P04629 1/20 0.32
LCK P06239 1/20 0.32
CSF1R P07333 1/20 0.32
RET P07949 1/20 0.32
MET P08581 1/20 0.32
PDGFRB P09619 1/20 0.32
PIM1 P11309 1/20 0.32
PDGFRA P16234 1/20 0.32
FLT3 P36888 1/20 0.32
MAPK8 P45983 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9245099 0.89 MCHR1 (0.41) GRM5EGLN1PTGESCHRNB2CHRNA2
SCHEMBL9246659 0.89 GRM2 (0.38) GRM5EGLN1PTGESCHRNB2CHRNA2
SCHEMBL9247860 0.87 CHRNB2 (0.33) GRM5EGLN1CHRNB2CHRNA2CHRNB4
SCHEMBL9245765 0.86 FFAR1 (0.38)
SCHEMBL9245211 0.86 PTGES (0.37) GRM5EGLN1PTGESCHRNB2CHRNA2
SCHEMBL9245001 0.85 GRM5 (0.46) GRM5EGLN1PTGESAURKAABL1
SCHEMBL9245011 0.85 GRM5 (0.46) GRM5EGLN1PTGESAURKAABL1
SCHEMBL9241425 0.83 GRM5 (0.45) GRM5EGLN1PTGESAURKAABL1
SCHEMBL9241419 0.83 GRM5 (0.45) GRM5EGLN1PTGESAURKAABL1
SCHEMBL9246583 0.83 GRM5 (0.45) GRM5EGLN1PTGESAURKAABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5447657-A Liquid crystal compounds HOFFMANN-LA ROCHE INC. (US) 1995-09-05 US disclosed