SCHEMBL9249093

SCHEMBL9249093

COc1ccc2c(c1)C(CCCCl)=CCC2

nearest known ligand 0.58

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.58
ABCB1 P08183 3/20 0.58
MPO P05164 1/20 0.51
MTNR1B P49286 3/20 0.43
NQO2 P16083 2/20 0.43
MTNR1A P48039 2/20 0.43
ALOX5 P09917 1/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16387896 0.91 SIGMAR1 (0.54) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL7784806 0.86 SIGMAR1 (0.58) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL7779874 0.86 SIGMAR1 (0.58) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL7779938 0.84 SIGMAR1 (0.57) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL1289512 0.82 SIGMAR1 (0.54) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL7780002 0.82 SIGMAR1 (0.55) SIGMAR1ABCB1MPOMTNR1BNQO2
Hydrochloric Acid SCHEMBL1289495 0.81 SIGMAR1 (0.53) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL13937830 0.80 MPO (0.77) SIGMAR1ABCB1MPOMTNR1BNQO2
SCHEMBL7787100 0.78 MTNR1A (0.54) SIGMAR1ABCB1MTNR1BNQO2MTNR1A
Hydrochloric Acid SCHEMBL11078947 0.78 MPO (0.55) SIGMAR1ABCB1MPOMTNR1BNQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0647222-A1 N(HETERO)-ARYL-N(HETERO)-TETRALIN-ALKYL-PIPERAZINE HAVING SEROTONINERGIC, DOPAMINERGIC AND ADRENERGIC ACTIVITY PHARMACIA & UPJOHN S.p.A. (IT) 1995-04-12 EP disclosed
WO-1994000441-A1 N(HETERO)-ARYL-N(HETERO)-TETRALIN-ALKYL-PIPERAZINE HAVING SEROTONINERGIC, DOPAMINERGIC AND ADRENERGIC ACTIVITY FARMITALIA CARLO ERBA S.R.L. (IT) 1994-01-06 WO disclosed