SCHEMBL9252364

SCHEMBL9252364

C=CCCc1cnc(-c2ccc(-c3ccc(F)c(F)c3)cc2)nc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.41
CYP11B2 P19099 2/20 0.41
CYP17A1 P05093 1/20 0.41
GRIN2B Q13224 14/20 0.38
GRIN1 Q05586 10/20 0.38
PDGFRB P09619 1/20 0.35
PDGFRA P16234 1/20 0.35
RARB P10826 1/20 0.33
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TP53 P04637 1/20 0.32
PKM P14618 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9249705 0.94 CYP11B1 (0.36) CYP11B1CYP11B2CYP17A1GRIN2BGRIN1
SCHEMBL9251920 0.92 CYP11B1 (0.39) CYP11B1CYP11B2CYP17A1GRIN2BGRIN1
SCHEMBL9253948 0.86 RARB (0.35) CYP11B1CYP11B2CYP17A1GRIN2BGRIN1
SCHEMBL9406468 0.83 RARB (0.36) CYP11B1CYP11B2GRIN2BPDGFRBPDGFRA
SCHEMBL9149216 0.81 RAB9A (0.49) CYP11B1CYP11B2CYP17A1GRIN2BGRIN1
SCHEMBL9250325 0.81 MAOB (0.46) HSD17B10
SCHEMBL9252692 0.80 SMN1; SMN2 (0.37) RARBNPC1RAB9ASMN1; SMN2HSD17B10
SCHEMBL9353374 0.79 CYP11B1 (0.38) CYP11B1CYP11B2CYP17A1GRIN2BGRIN1
SCHEMBL15783706 0.77 RARB (0.57) CYP11B1CYP11B2CYP17A1RARBNPC1
SCHEMBL9252022 0.77 RARB (0.40) GRIN2BRARBNPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
EP-0315014-B1 Halogenated benzene derivatives HOFFMANN LA ROCHE (CH) 1994-01-12 EP disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
EP-0315014-A2 Halogenated benzene derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed