SCHEMBL9249705

SCHEMBL9249705

C=CCCc1cnc(-c2ccc(F)c(F)c2)nc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
CYP17A1 P05093 1/20 0.36
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
GPR68 Q15743 1/20 0.34
GRIN2B Q13224 4/20 0.34
GRIN1 Q05586 3/20 0.34
NPC1 O15118 1/20 0.33
TP53 P04637 1/20 0.33
PKM P14618 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
NOTUM Q6P988 1/20 0.32
GRM2 Q14416 1/20 0.32
RARB P10826 1/20 0.31
FYN P06241 1/20 0.31
NPY5R Q15761 1/20 0.31
CHRNB2 P17787 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252364 0.94 CYP11B1 (0.41) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9253948 0.91 RARB (0.35) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9251920 0.86 CYP11B1 (0.39) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9353374 0.84 CYP11B1 (0.38) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9406468 0.83 RARB (0.36) CYP11B1CYP11B2PDGFRBPDGFRAGRIN2B
SCHEMBL7519352 0.80 RAB9A (0.51) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9252692 0.80 SMN1; SMN2 (0.37) NPC1RAB9ASMN1; SMN2HSD17B10NOTUM
SCHEMBL12357413 0.79 ALOX5AP (0.39) GRM2
SCHEMBL9646838 0.78 GRIN2B (0.34) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA
SCHEMBL9646834 0.78 GRIN2B (0.34) CYP11B1CYP11B2CYP17A1PDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5454974-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1995-10-03 US disclosed
US-5302317-A Halobenzene liquid crystals HOFFMANN-LA ROCHE INC. (US) 1994-04-12 US disclosed
EP-0315014-B1 Halogenated benzene derivatives HOFFMANN LA ROCHE (CH) 1994-01-12 EP disclosed
US-5230826-A HALOBENZENE LIQUID CRYSTALS HOFFMANN-LA ROCHE INC. (US) 1993-07-27 US disclosed
EP-0315014-A2 Halogenated benzene derivatives F. HOFFMANN-LA ROCHE AG (CH) 1989-05-10 EP disclosed