SCHEMBL9250622

SCHEMBL9250622

COC1C(Cn2cncn2)C(OCc2ccc3ccccc3n2)CCC1(C)C

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.34
HCRTR1 O43613 5/20 0.33
HCRTR2 O43614 5/20 0.33
PDE10A Q9Y233 4/20 0.33
ALOX5AP P20292 4/20 0.33
CYP1A2 P05177 3/20 0.33
CYSLTR2 Q9NS75 1/20 0.32
CYSLTR1 Q9Y271 1/20 0.32
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9250615 1.00 REN (0.34) RENHCRTR1HCRTR2PDE10AALOX5AP
SCHEMBL9245399 0.91 REN (0.34) RENHCRTR1HCRTR2PDE10ACYP1A2
SCHEMBL9242863 0.84 CYP1A2 (0.35) RENHCRTR1HCRTR2PDE10ACYP1A2
SCHEMBL9244604 0.84 CALCA (0.36) HCRTR1HCRTR2PDE10AALOX5APCYSLTR2
SCHEMBL9244600 0.84 CALCA (0.36) HCRTR1HCRTR2PDE10AALOX5APCYSLTR2
SCHEMBL9244509 0.83 GAA (0.38) RENHCRTR1HCRTR2
SCHEMBL9244519 0.83 GAA (0.38) RENHCRTR1HCRTR2
SCHEMBL9245404 0.82
SCHEMBL9244554 0.82 ALOX5AP (0.38) ALOX5APCYSLTR2CYSLTR1BRD4
SCHEMBL8715857 0.82 ALOX5AP (0.38) ALOX5APCYSLTR2CYSLTR1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5449785-A Fungicides with triazole groups HOFFMANN-LA ROCHE INC. (US) 1995-09-12 US disclosed
EP-0524439-A1 Novel cyclohexane and tetrahydropyran derivatives and antifungal compositions containing these derivatives F.HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT (CH) 1993-01-27 EP disclosed