SCHEMBL8715857

SCHEMBL8715857

COC1C(CO)C(OCc2ccc3ccccc3n2)CCC1(C)C

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 11/20 0.38
CYSLTR1 Q9Y271 4/20 0.38
CYSLTR2 Q9NS75 1/20 0.37
GPBAR1 Q8TDU6 2/20 0.36
BRD4 O60885 1/20 0.36
ALOX5 P09917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9244554 1.00 ALOX5AP (0.38) ALOX5APCYSLTR1CYSLTR2GPBAR1BRD4
SCHEMBL8719748 0.90 CYP1A2 (0.35) ALOX5APCYSLTR1ALOX5
SCHEMBL9244570 0.90 CYP1A2 (0.35) ALOX5APCYSLTR1ALOX5
SCHEMBL9250615 0.82 REN (0.34) ALOX5APCYSLTR1CYSLTR2BRD4
SCHEMBL9244604 0.82 CALCA (0.36) ALOX5APCYSLTR1CYSLTR2BRD4
SCHEMBL9250622 0.82 REN (0.34) ALOX5APCYSLTR1CYSLTR2BRD4
SCHEMBL9244600 0.82 CALCA (0.36) ALOX5APCYSLTR1CYSLTR2BRD4
SCHEMBL9244571 0.79 ALDH1A1 (0.34) ALOX5AP
SCHEMBL8717311 0.78 PDE10A (0.36) ALOX5APCYSLTR1CYSLTR2ALOX5
SCHEMBL8714319 0.77 ALOX5AP (0.35) ALOX5APCYSLTR1CYSLTR2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719291-A FUNGICIDE HOFFMANN-LA ROCHE INC. (US) 1998-02-17 US disclosed
US-5449785-A Fungicides with triazole groups HOFFMANN-LA ROCHE INC. (US) 1995-09-12 US disclosed
EP-0524439-A1 Novel cyclohexane and tetrahydropyran derivatives and antifungal compositions containing these derivatives F.HOFFMANN-LA ROCHE & CO. AKTIENGESELLSCHAFT (CH) 1993-01-27 EP disclosed