SCHEMBL9251368

SCHEMBL9251368

Cc1ccc(-c2nc3cc(C(=O)NCCC(=O)O)ccc3n2C)c(C(=N)N)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 6/20 0.45
HDAC1 Q13547 3/20 0.45
HDAC8 Q9BY41 3/20 0.45
ITGB3 P05106 2/20 0.44
ITGA2B P08514 2/20 0.44
HDAC3 O15379 2/20 0.43
HDAC2 Q92769 2/20 0.43
F2 P00734 6/20 0.42
ATM Q13315 1/20 0.41
NAMPT P43490 1/20 0.40
GCG P01275 1/20 0.40
MAPK10 P53779 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9248587 0.91 HDAC6 (0.43) HDAC6HDAC1HDAC8HDAC3HDAC2
SCHEMBL9249002 0.87 ITGB3 (0.50) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9256145 0.85 F2 (0.49) ITGB3ITGA2BF2
SCHEMBL9248855 0.84 ITGB3 (0.47) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9249490 0.84 HDAC1 (0.56) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9254163 0.83 KDM4E (0.41) HDAC6HDAC1HDAC8HDAC3HDAC2
SCHEMBL9257024 0.81 KDM4E (0.41) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9255028 0.80 ITGB3 (0.47) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9254680 0.79 HPGD (0.45) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9245467 0.78 HDAC1 (0.38) HDAC6HDAC1HDAC8HDAC3HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed