SCHEMBL9254680

SCHEMBL9254680

CCCCNC(=N)c1ccccc1-c1nc2cc(C(=O)NCCC(=O)O)ccc2n1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.45
TP53 P04637 2/20 0.45
HDAC6 Q9UBN7 3/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC8 Q9BY41 1/20 0.44
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
POLB P06746 1/20 0.42
ALOX15 P16050 1/20 0.42
CASP1 P29466 1/20 0.42
BLM P54132 1/20 0.42
CASP7 P55210 1/20 0.42
MCL1 Q07820 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42
MRGPRX1 Q96LB2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251757 0.92 HPGD (0.44) HPGDTP53HDAC6HDAC1HDAC8
SCHEMBL9251368 0.79 HDAC6 (0.45) TP53HDAC6HDAC1HDAC8ATM
SCHEMBL9249002 0.77 ITGB3 (0.50) HDAC6HDAC1HDAC8ITGB3ITGA2B
SCHEMBL9251361 0.76 HDAC6 (0.55) TP53HDAC6HDAC1HDAC8MAPT
SCHEMBL9256145 0.75 F2 (0.49) ITGB3ITGA2B
SCHEMBL9249490 0.75 HDAC1 (0.56) HDAC6HDAC1HDAC8PTGER4NAMPT
SCHEMBL9248855 0.74 ITGB3 (0.47) HPGDHDAC6HDAC1HDAC8ALDH1A1
SCHEMBL9249572 0.73 ITGB3 (0.56) HDAC6HDAC1HDAC8PTGER4NAMPT
SCHEMBL9251208 0.73 ITGB3 (0.53) PTGER4ITGB3ITGA2B
SCHEMBL9255028 0.72 ITGB3 (0.47) HDAC6HDAC1HDAC8NAMPTITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed