SCHEMBL9251487

SCHEMBL9251487

CC1=N[C@@H](NC(=O)Nc2cccc(-c3nnn[nH]3)c2)C(=O)N(C)c2ccccc21

nearest known ligand 0.62

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 18/20 0.62
KCNH2 Q12809 1/20 0.60
CCKAR P32238 4/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8542118 0.91 CCKBR (0.77) CCKBRKCNH2CCKAR
SCHEMBL9699970 0.87 CCKBR (0.71) CCKBR
SCHEMBL9303173 0.86 CCKBR (0.71) CCKBR
SCHEMBL9422497 0.86 CCKBR (0.53) CCKBRKCNH2CCKAR
SCHEMBL8543069 0.81 CCKBR (0.62) CCKBRKCNH2CCKAR
SCHEMBL8546195 0.80 CCKBR (0.64) CCKBRKCNH2CCKAR
SCHEMBL8547291 0.80 CCKBR (0.62) CCKBRCCKAR
SCHEMBL9545575 0.79 CCKBR (0.74) CCKBRKCNH2CCKAR
SCHEMBL8540475 0.79 CCKBR (0.51) CCKBRCCKAR
SCHEMBL9573642 0.79 CCKBR (0.62) CCKBRKCNH2CCKAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5451582-A Cholecystokinins and gastrin receptor antagonists MERCK SHARP & DOHME LTD. (GB) 1995-09-19 US claimed
WO-1993017011-A1 BENZODIAZEPINE DERIVATIVES, AS CCK AND GASTRIN ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1993-09-02 WO claimed
US-5451582-A Cholecystokinins and gastrin receptor antagonists MERCK SHARP & DOHME LTD. (GB) 1995-09-19 US disclosed