SCHEMBL9252897

SCHEMBL9252897

O=C(CCCC1CCN(Cc2ccccc2)CC1)c1ccc(N2CCCC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 6/20 0.67
BCHE P06276 3/20 0.67
FAAH O00519 1/20 0.57
HTR1A P08908 1/20 0.56
SLC6A4 P31645 1/20 0.56
CHRM4 P08173 1/20 0.55
HTR2A P28223 1/20 0.55
HTR2C P28335 1/20 0.55
HTR2B P41595 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253392 0.97 ACHE (0.65) ACHEBCHEFAAHHTR1ASLC6A4
Fumaric Acid SCHEMBL9254343 0.95 ACHE (0.60) ACHEBCHEFAAHHTR1ASLC6A4
Fumaric Acid SCHEMBL9254339 0.95 ACHE (0.60) ACHEBCHEFAAHHTR1ASLC6A4
SCHEMBL4500124 0.93 ACHE (0.77) ACHEBCHEHTR1ASLC6A4
Fumaric Acid SCHEMBL9249220 0.92 ACHE (0.59) ACHEBCHEFAAHHTR1ASLC6A4
Fumaric Acid SCHEMBL9249239 0.92 ACHE (0.59) ACHEBCHEFAAHHTR1ASLC6A4
SCHEMBL9246613 0.86 HTR2A (0.59) ACHEBCHEHTR2AHTR2CHTR2B
SCHEMBL9253116 0.85 ACHE (0.71) ACHEBCHEFAAHCHRM4
SCHEMBL7806521 0.83 ACHE (0.71) ACHEBCHEFAAH
SCHEMBL9254685 0.82 ACHE (0.60) ACHEBCHEHTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed