SCHEMBL9253425

SCHEMBL9253425

O=c1[nH]c(=O)c2[nH]c(-c3cccs3)nc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 2/20 0.59
KDM4E B2RXH2 4/20 0.51
HPGD P15428 4/20 0.51
PKM P14618 1/20 0.51
ALDH1A1 P00352 3/20 0.49
MAPK1 P28482 2/20 0.49
HTT P42858 2/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
GLA P06280 1/20 0.49
GAA P10253 1/20 0.49
MAPT P10636 1/20 0.49
ERCC1 P07992 6/20 0.48
FEN1 P39748 6/20 0.48
ERCC4 Q92889 6/20 0.48
TYMP P19971 1/20 0.48
DNASE1 P24855 1/20 0.47
ADORA3 P0DMS8 1/20 0.46
ADORA2A P29274 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378879 0.74 ADORA2B (1.00) ADORA2BHPGDALDH1A1KMT2AMEN1
SCHEMBL6783434 0.71 GRIA1 (0.59) ADORA2BKDM4EHPGDPKMALDH1A1
SCHEMBL18036538 0.70 ADORA2B (0.63) ADORA2BKDM4EHPGDPKMALDH1A1
SCHEMBL4400471 0.70 HPGD (0.51) KDM4EHPGDPKMALDH1A1GAA
SCHEMBL23607984 0.69 ADORA2B (0.71) ADORA2BKDM4EHPGDALDH1A1MAPK1
SCHEMBL4927186 0.69 ADORA2B (0.70) ADORA2BKDM4EHPGDALDH1A1KMT2A
SCHEMBL11830857 0.68 HPGD (1.00) KDM4EHPGDPKMALDH1A1MAPK1
SCHEMBL30362164 0.68 HPGD (1.00) KDM4EHPGDPKMALDH1A1MAPK1
SCHEMBL42351 0.68 NOS1 (0.55) ADORA2BKDM4EHPGDPKMALDH1A1
SCHEMBL1051055 0.68 ADORA2B (0.60) ADORA2BKDM4EHPGDALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103254194-B Preparation method of 8-thiaxanthine compound UNIV ZHEJIANG NORMAL 2015-07-08 CN disclosed
CN-103275079-B Preparation method for 8-aryl or vinyl-substituted xanthine compound UNIV ZHEJIANG NORMAL 2015-06-24 CN disclosed
CN-103275079-A Preparation method for 8-aryl or vinyl-substituted xanthine compound UNIV ZHEJIANG NORMAL 2013-09-04 CN disclosed
CN-103254194-A Preparation method of 8-thiaxanthine compound UNIV ZHEJIANG NORMAL 2013-08-21 CN disclosed
US-5453426-A Sulfur-containing xanthine derivatives as adenosine antagonists THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-09-26 US disclosed
WO-1990012797-A1 SULFER-CONTAINING XANTHINE DERIVATIVES AS ADENOSIN ANTAGONISTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1990-11-01 WO disclosed