SCHEMBL9253489

SCHEMBL9253489

CN(C)c1ccc(CC2CCN(C(=O)c3ccccc3)CC2)cc1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.58
CA12 O43570 1/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA14 Q9ULX7 1/20 0.58
GAA P10253 1/20 0.58
CYP2C9 P11712 4/20 0.56
CYP2C19 P33261 4/20 0.56
MAPK14 Q16539 4/20 0.56
HTR2B P41595 2/20 0.56
ACHE P22303 1/20 0.54
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7241024 0.95 HTT (0.65) HTTCA12CA1CA2CA7
SCHEMBL7242121 0.86 LMNA (0.58) HTTCA12CA1CA2CA7
SCHEMBL7232379 0.86 HTT (0.73) HTTCA12CA1CA2CA7
SCHEMBL9247360 0.84 CCR5 (0.49) CYP2C9CYP2C19MAPK14HTR2BMEN1
SCHEMBL10719972 0.83 HTT (0.78) HTTCA12CA1CA2CA7
SCHEMBL13108352 0.83 CYP2C9 (0.64) HTTCA12CA1CA2CA7
SCHEMBL29941294 0.80 HTT (0.69) HTTCA12CA1CA2CA7
SCHEMBL10723602 0.80 MGLL (0.67) HTTCA12CA1CA2CA7
SCHEMBL5366293 0.79 HTT (0.67) HTTCA12CA1CA2CA7
SCHEMBL1720920 0.79 MGLL (0.69) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed