SCHEMBL9253975

SCHEMBL9253975

COC(=O)CCc1ccc(-n2nnc(-c3ccc(C#N)cc3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
CHRNB2 P17787 1/20 0.47
CHRNA5 P30532 1/20 0.47
CHRNA4 P43681 1/20 0.47
MAPT P10636 3/20 0.43
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
AOC3 Q16853 2/20 0.41
S1PR1 P21453 2/20 0.41
S1PR5 Q9H228 2/20 0.41
ABCG2 Q9UNQ0 5/20 0.41
MMP9 P14780 2/20 0.40
POLB P06746 1/20 0.39
ABCB1 P08183 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9251339 0.83 HPGD (0.49) HPGDTSHRHSD17B10MAPTTP53
Hydrochloric Acid SCHEMBL9254302 0.82 HPGD (0.48) HPGDTSHRHSD17B10MAPTTP53
SCHEMBL3628694 0.80 CYP11B1 (0.56) HPGDTSHRHSD17B10CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL3628690 0.79 CYP11B1 (0.55) HPGDTSHRHSD17B10CYP11B1CYP11B2
SCHEMBL1338556 0.79 CYP11B1 (0.60) CYP11B1CYP11B2MAPTPOLBALDH1A1
SCHEMBL10664707 0.79 CHRNB2 (0.69) CHRNB2CHRNA5CHRNA4MAPTAOC3
SCHEMBL9256828 0.78 TSHR (0.68) HPGDTSHRHSD17B10MAPTTP53
SCHEMBL9251061 0.77 CYP11B1 (0.52) CYP11B1CYP11B2MAPTS1PR1POLB
SCHEMBL9251931 0.77 CYP11B1 (0.52) HPGDHSD17B10CYP11B1CYP11B2MAPT
SCHEMBL9259632 0.74 CYP11B1 (0.47) HPGDCYP11B1CYP11B2MAPTS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed