SCHEMBL9254097

SCHEMBL9254097

Oc1c(-c2cccc(F)c2)cnc2c(-c3cc(-c4ccccc4)cs3)cnn12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.39
RAB9A P51151 5/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
RXFP1 Q9HBX9 2/20 0.38
EGLN2 Q96KS0 1/20 0.34
FYN P06241 2/20 0.34
HSD17B1 P14061 3/20 0.34
HSD17B2 P37059 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPT P10636 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KDR P35968 3/20 0.33
LCK P06239 2/20 0.33
HCK P08631 2/20 0.33
SRC P12931 2/20 0.33
HPGDS O60760 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688673 0.90 NPC1 (0.47) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9169606 0.90 RAB9A (0.47) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9172844 0.89 HSD17B1 (0.46) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9173628 0.89 RAB9A (0.45) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9168612 0.86 NPC1 (0.39) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9165874 0.86 HSD17B1 (0.44) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9168862 0.85 NPC1 (0.39) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9170467 0.85 KDR (0.46) NPC1RAB9AMEN1KMT2AEGLN2
SCHEMBL9166749 0.84 RAB9A (0.41) NPC1RAB9AMEN1KMT2ARXFP1
SCHEMBL9173884 0.84 RAB9A (0.40) NPC1RAB9AMEN1KMT2ARXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5420128-A Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-05-30 US disclosed
EP-0503099-A1 PYRIMIDINE DERIVATIVE, PRODUCTION THEREOF, AND ANDROGEN INHIBITOR OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-09-16 EP disclosed