SCHEMBL9254441

SCHEMBL9254441

CCCC(=O)OCOC(=O)CCc1ccc(-c2nc(-c3cccc(C(=O)OCc4ccccc4)c3C(=N)N)cn2C)cc1

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.35
MAPK1 P28482 2/20 0.35
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
DHODH Q02127 3/20 0.35
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
PARP1 P09874 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
CYP3A4 P08684 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CASP3 P42574 1/20 0.35
RAB9A P51151 1/20 0.35
SENP8 Q96LD8 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254434 0.94 KDM4E (0.35) TSHRMAPK1ALDH1A1KDM4EHPGD
SCHEMBL9254565 0.92 PARP1 (0.34) TSHRMAPK1ALDH1A1KDM4EHPGD
SCHEMBL9254562 0.86 PARP1 (0.34) TSHRMAPK1ALDH1A1KDM4EHPGD
SCHEMBL9255731 0.80 ALDH1A1 (0.38) TSHRALDH1A1KDM4EHPGDDHODH
SCHEMBL9255106 0.79 ALDH1A1 (0.36) TSHRALDH1A1KDM4EHPGDDHODH
SCHEMBL9253893 0.78 F10 (0.40) TSHRRAB9A
SCHEMBL9247338 0.76 MAPT (0.38) TSHRALDH1A1KDM4EHPGDDHODH
SCHEMBL9253869 0.75 F2 (0.40) ALDH1A1KDM4EHPGDADORA2AADORA1
SCHEMBL9256887 0.74 ALDH1A1 (0.37) TSHRALDH1A1KDM4EHPGDL3MBTL1
SCHEMBL9288922 0.73 TDP1 (0.43) ALDH1A1KDM4EL3MBTL1TDP1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed