SCHEMBL9256887

SCHEMBL9256887

CCOC(=O)OC(C)OC(=O)CCc1ccc(-c2nc(-c3ccc(C(=O)OCc4ccccc4)cc3C(=N)N)cn2C)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
MAPT P10636 7/20 0.37
NPC1 O15118 3/20 0.34
RAB9A P51151 3/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
POLB P06746 1/20 0.34
LMNA P02545 1/20 0.34
F2 P00734 1/20 0.33
NAMPT P43490 2/20 0.32
F10 P00742 1/20 0.32
JMJD6 Q6NYC1 1/20 0.32
PTPN1 P18031 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PCSK9 Q8NBP7 1/20 0.31
DGAT1 O75907 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257668 0.90 KDM4E (0.36) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9247338 0.87 MAPT (0.38) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9255731 0.86 ALDH1A1 (0.38) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9255106 0.84 ALDH1A1 (0.36) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9255799 0.82 F10 (0.41) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL9256883 0.81 KDM4E (0.36) ALDH1A1KDM4EHPGDMAPTNPC1
SCHEMBL9253103 0.81 ALOX5 (0.38) ALDH1A1KDM4EHPGDMAPTF2
SCHEMBL9257625 0.79 MAPT (0.33) ALDH1A1MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL9257107 0.78 F2 (0.37) ALDH1A1HPGDRAB9AF2F10
SCHEMBL9254257 0.76 HDAC1 (0.33) ALDH1A1KDM4EHPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed