SCHEMBL9254481

SCHEMBL9254481

CNc1ccc(Sc2cccc(Br)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 4/20 0.40
ALDH1A1 P00352 2/20 0.38
MAPT P10636 1/20 0.38
APP P05067 1/20 0.38
EGFR P00533 3/20 0.38
EPHB2 P29323 1/20 0.38
ERBB2 P04626 1/20 0.38
MAOB P27338 3/20 0.37
TYMS P04818 2/20 0.36
MAPK1 P28482 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
TSHR P16473 1/20 0.35
GRM5 P41594 1/20 0.35
PLK4 O00444 1/20 0.35
PTGIR P43119 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11819273 0.81 MAOA (0.50) MAOAALDH1A1MAOBMAPK1GRM5
SCHEMBL31337906 0.80 MAOA (0.48) MAOAALDH1A1MAOBTYMSMAPK1
SCHEMBL3289392 0.80 MAOA (0.48) MAOAALDH1A1MAOBTYMSMAPK1
SCHEMBL29543964 0.80 MAOA (0.48) MAOAALDH1A1MAOBTYMSMAPK1
SCHEMBL17643520 0.79 ALDH1A1 (0.50) MAOAALDH1A1MAPTMAOBTYMS
SCHEMBL8953701 0.79 IDO1 (0.51) ALDH1A1MAPTEGFRMTNR1AMTNR1B
SCHEMBL3285262 0.78 HTR2C (0.47) MAOAALDH1A1MAPTMAOBMAPK1
SCHEMBL30385602 0.78 HTR2C (0.47) MAOAALDH1A1MAPTMAOBMAPK1
SCHEMBL6975747 0.78 TSHR (0.59) MAOAALDH1A1MAPTAPPMAOB
SCHEMBL10595966 0.78 MAOA (0.47) MAOAALDH1A1MAOBTYMSMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5432194-A Antiallergens, antinflammatory agents ABBOTT LABORATORIES (US) 1995-07-11 US disclosed
WO-1994026264-A1 (4-ALKOXYPYRAN-4-YL) SUBSTITUTED ARYLALKYLARYL-, ARYLALKENYLARYL-, AND ARYLALKYNYLARYLUREA INHIBITORS OF 5-LIPOXYGENASE ABBOTT LABORATORIES (US) 1994-11-24 WO disclosed