SCHEMBL9254542

SCHEMBL9254542

N#Cc1ccc(-c2ccc(-c3nnn[nH]3)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP3 P08254 1/20 0.44
NOTUM Q6P988 2/20 0.41
CYP11B2 P19099 1/20 0.41
KIF11 P52732 2/20 0.40
RHEB Q15382 1/20 0.40
DGAT1 O75907 1/20 0.38
SOAT1 P35610 1/20 0.38
KCNH2 Q12809 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
RIPK1 Q13546 1/20 0.37
IDO1 P14902 1/20 0.37
MAPK13 O15264 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4402319 0.98 NOTUM (0.42) MMP3NOTUMCYP11B2KIF11RHEB
SCHEMBL13411813 0.84 ADH5 (0.36)
SCHEMBL12536128 0.84 CLK4 (0.45) NOTUMGABRA1GABRG2GABRB3GABRA5
SCHEMBL2028396 0.82 ADH5 (0.32)
SCHEMBL18424351 0.79 KEAP1 (0.37) CA12CA1CA2CA9MAPK14
SCHEMBL17254440 0.78 ESR1 (0.33)
SCHEMBL5784940 0.77 CLK4 (0.49) NOTUMGABRA1GABRG2GABRB3GABRA5
SCHEMBL27513088 0.77
SCHEMBL6505461 0.76 NR1H2 (0.41) DGAT1MAPK13MAPK12MAPK11MAPK14
SCHEMBL6879531 0.75 KDM4E (0.48) MMP3MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed