SCHEMBL9254545

SCHEMBL9254545

COC1CCOC(c2cccc(COc3ccc4c(-c5ccccc5)cc(=O)oc4c3)c2)C1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.61
ALDH1A1 P00352 2/20 0.48
HPGD P15428 2/20 0.48
USP2 O75604 1/20 0.48
NPC1 O15118 3/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RAB9A P51151 2/20 0.47
MAOA P21397 1/20 0.47
CASP3 P42574 1/20 0.47
SENP8 Q96LD8 1/20 0.47
SENP7 Q9BQF6 1/20 0.47
SENP6 Q9GZR1 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
AR P10275 2/20 0.45
CA12 O43570 1/20 0.45
CA9 Q16790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9267747 0.90 MAOB (0.48) MAOBNPC1RAB9AMAOACASP3
SCHEMBL9258559 0.90 MAOB (0.48) MAOBNPC1RAB9AMAOACASP3
SCHEMBL9265290 0.90 MAOB (0.63) MAOBALDH1A1HPGDUSP2NPC1
SCHEMBL9259277 0.88 RAB9A (0.61) MAOBNPC1RAB9AMAOACASP3
SCHEMBL9267165 0.85 KMT2A (0.51) MAOBALDH1A1HPGDNPC1CYP2C9
SCHEMBL9263722 0.84 NPC1 (0.58) MAOBNPC1RAB9AMAOAMEN1
SCHEMBL9161622 0.84 MAOB (0.39) MAOBALDH1A1HPGDNPC1SMN1; SMN2
SCHEMBL9158135 0.83 ALOX5 (0.42) MAOBALDH1A1HPGDNPC1SMN1; SMN2
SCHEMBL9154816 0.83 MAOB (0.38) MAOBALDH1A1HPGDNPC1SMN1; SMN2
SCHEMBL9263552 0.83 MAOB (0.47) MAOBNPC1RAB9AMAOAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424320-A Antihistamine, antiallergic, antiinflammatory and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1995-06-13 US disclosed
US-5360815-A Heteroaryl cinnamic acids as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1994-11-01 US disclosed