SCHEMBL9255562

SCHEMBL9255562

CC(=O)N1CCC(C(c2ccccc2)N2CCN(Cc3ccccc3)CC2)CC1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.54
CACNA2D1 P54289 4/20 0.54
CACNA1B Q00975 4/20 0.54
CACNB1 Q02641 4/20 0.54
CACNA1C Q13936 3/20 0.54
CYP2D6 P10635 1/20 0.53
ALDH1A1 P00352 2/20 0.51
SCN5A Q14524 1/20 0.51
SCN9A Q15858 1/20 0.51
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
HRH3 Q9Y5N1 1/20 0.49
MAOB P27338 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
POLB P06746 1/20 0.47
RAB9A P51151 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2791280 0.84 CACNA2D1 (0.66) CACNA2D1CACNA1BCACNB1CACNA1CCYP2D6
SCHEMBL20804559 0.82 ATM (0.54) ATMALDH1A1SCN5ASCN9AKMT2A
SCHEMBL20804476 0.81 ATM (0.52) ATMALDH1A1SCN5ASCN9AKMT2A
SCHEMBL8211709 0.81 CACNA2D1 (0.53) CACNA2D1CACNA1BCACNB1CACNA1CCYP2D6
SCHEMBL3398020 0.80 CACNA2D1 (0.56) ATMCACNA2D1CACNA1BCACNB1CACNA1C
Hydrochloric Acid SCHEMBL27266176 0.79 CACNA2D1 (0.57) CACNA2D1CACNA1BCACNB1CACNA1CCYP2D6
SCHEMBL1943497 0.79 HRH3 (0.75) ATMCYP2D6ALDH1A1KMT2AMEN1
SCHEMBL7501907 0.76 ABL1 (0.54) ATMKMT2AMEN1
SCHEMBL26358318 0.76 OPRM1 (0.50) ATMALDH1A1KMT2AMEN1
SCHEMBL26358315 0.76 LMNA (0.56) CYP2D6ALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed