SCHEMBL9255900

SCHEMBL9255900

COC(=O)CCc1ccc(-c2nc(-c3ccc(C4(N)CC4)cc3)cn2C)cc1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AKT2 P31751 10/20 0.49
AKT1 P31749 9/20 0.49
HRH3 Q9Y5N1 4/20 0.41
SYK P43405 2/20 0.37
KIT P10721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257888 0.96 AKT2 (0.51) AKT2AKT1HRH3
SCHEMBL9254431 0.89 AKT2 (0.44) AKT2AKT1HRH3SYK
SCHEMBL9248511 0.85 HRH3 (0.42) HRH3SYK
SCHEMBL9251212 0.85 HRH3 (0.42) HRH3
SCHEMBL9259539 0.84 AKT2 (0.47) AKT2AKT1HRH3
SCHEMBL9250844 0.82 HRH3 (0.42) HRH3
SCHEMBL9257434 0.81 NPC1 (0.42) HRH3
SCHEMBL9259602 0.81 HRH3 (0.40) HRH3SYK
SCHEMBL9255567 0.81 HRH3 (0.40) HRH3SYK
SCHEMBL9259034 0.81 NPC1 (0.42) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
US-5401768-A Prostaglandin derivative, antiulcer, hypotensive, anticoagulant TORAY INDUSTRIES, INC. (JP) 1995-03-28 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed