SCHEMBL9256586

SCHEMBL9256586

CCP(=O)(CC)c1ccc(-c2cn(C)c(-c3ccc(CCC(=O)OC)cc3)n2)c(C(=N)N)c1

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
HRH3 Q9Y5N1 1/20 0.33
PTPN1 P18031 2/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CCR9 P51686 2/20 0.31
VDR P11473 1/20 0.31
PPARD Q03181 1/20 0.31
SYK P43405 1/20 0.30
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257107 0.85 F2 (0.37) HDAC1HRH3HPGDTSHRHSD17B10
SCHEMBL9254257 0.80 HDAC1 (0.33) HDAC1HRH3HPGDTSHRHSD17B10
SCHEMBL9259034 0.78 NPC1 (0.42) HRH3HPGDTSHRHSD17B10
SCHEMBL9257434 0.78 NPC1 (0.42) HRH3HPGDTSHRHSD17B10
Hydrochloric Acid SCHEMBL9256062 0.77 NPC1 (0.41) HRH3HPGDTSHRHSD17B10
SCHEMBL9253103 0.77 ALOX5 (0.38) HPGD
SCHEMBL9256582 0.74 HRH3 (0.36) HDAC1HRH3HPGDTSHRHSD17B10
SCHEMBL9248511 0.73 HRH3 (0.42) HDAC1HRH3HPGDTSHRHSD17B10
SCHEMBL9251212 0.73 HRH3 (0.42) HDAC1HRH3HPGDTSHRHSD17B10
SCHEMBL9256832 0.72 ACVR1 (0.41) HRH3HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed