SCHEMBL9257637

SCHEMBL9257637

CC(=O)N1CCC(C(=O)c2ccc(N3CCNCC3)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 4/20 0.51
ALDH1A1 P00352 2/20 0.50
USP2 O75604 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CYP2D6 P10635 1/20 0.48
MGLL Q99685 3/20 0.47
POLB P06746 1/20 0.46
LMNA P02545 1/20 0.46
CASP6 P55212 1/20 0.46
GFER P55789 1/20 0.46
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
MAPT P10636 1/20 0.45
ACVR1 Q04771 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9255076 0.87 HSD11B1 (0.54) HSD11B1ALDH1A1TSHRHSD17B10MEN1
SCHEMBL9252527 0.86 HSD11B1 (0.53) HSD11B1ALDH1A1MEN1KMT2AMGLL
SCHEMBL9254041 0.86 HSD11B1 (0.53) HSD11B1ALDH1A1MEN1KMT2AMGLL
SCHEMBL9249192 0.85 HSD11B1 (0.69) HSD11B1ALDH1A1HSD17B10MEN1KMT2A
SCHEMBL10445779 0.78 KDM4E (0.46) ALDH1A1TSHRHSD17B10MEN1KMT2A
SCHEMBL29448588 0.78 KMT2A (0.77) HSD11B1ALDH1A1TSHRMEN1KMT2A
Hydrochloric Acid SCHEMBL9247465 0.77 KDM4E (0.48) ALDH1A1TSHRHSD17B10MEN1KMT2A
Hydrochloric Acid SCHEMBL9257378 0.77 MEN1 (0.60) HSD11B1ALDH1A1USP2TSHRHSD17B10
SCHEMBL13944269 0.77 MEN1 (0.54) HSD11B1ALDH1A1TSHRMEN1KMT2A
SCHEMBL14640729 0.77 MEN1 (0.56) HSD11B1ALDH1A1MEN1KMT2AMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5441967-A Treating cerebral edema; anticholinesterase or brain function-improving agent TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-08-15 US disclosed
US-5294625-A 1-benzyl,4-((4-dialkylaminophenyl)carbonyl)piperidines TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0378207-B1 CYCLIC AMINE COMPOUNDS AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 1993-09-22 EP disclosed
US-5177087-A Cerebral edema, cholinesterase inhibitor TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-05 US disclosed
EP-0378207-A1 Cyclic amine compounds and their use Takeda Chemical Industries, Ltd. (JP) 1990-07-18 EP disclosed