SCHEMBL9258181

SCHEMBL9258181

Cn1c(=O)c2c(nc(-c3cccs3)n2C)n(C)c1=O

nearest known ligand 0.68

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 4/20 0.61
ADORA2A P29274 4/20 0.61
MAOB P27338 2/20 0.56
GAA P10253 1/20 0.53
MAPT P10636 1/20 0.53
TP53 P04637 1/20 0.52
ERCC1 P07992 1/20 0.50
FEN1 P39748 1/20 0.50
ERCC4 Q92889 1/20 0.50
KDM4E B2RXH2 2/20 0.49
HSD17B10 Q99714 1/20 0.49
ADORA1 P30542 1/20 0.48
ALDH1A1 P00352 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
RXFP1 Q9HBX9 1/20 0.47
MAOA P21397 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9257945 0.86 ERCC1 (0.48) ADORA2BADORA2AMAOBGAAMAPT
SCHEMBL17626212 0.81 ALDH1A1 (0.56) ADORA2BADORA2AMAPTTP53ERCC1
SCHEMBL2403877 0.78 ADORA2B (0.69) ADORA2BADORA2AMAOBALDH1A1RXFP1
SCHEMBL4146728 0.76 ADORA2B (1.00) ADORA2BADORA2AMAOBALDH1A1SMN1; SMN2
SCHEMBL25089930 0.74 ADORA2B (0.65) ADORA2BADORA2AMAOBMAOA
SCHEMBL593805 0.73 ADORA2B (0.77) ADORA2BADORA2AMAOBTP53RXFP1
SCHEMBL28501882 0.72 ADORA1 (0.64) ADORA2BADORA2AKDM4EHSD17B10ADORA1
SCHEMBL1347557 0.71 ADORA2A (0.73) ADORA2BADORA2AMAOBMAOA
SCHEMBL7032893 0.70 ADORA2B (0.68) ADORA2BADORA2AMAOBKDM4EALDH1A1
SCHEMBL9118620 0.70 ALDH1A1 (0.49) MAPTTP53ERCC1FEN1ERCC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5453426-A Sulfur-containing xanthine derivatives as adenosine antagonists THE UNITED STATES OF AMERICA AS REPRESENTED BY THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1995-09-26 US disclosed
WO-1990012797-A1 SULFER-CONTAINING XANTHINE DERIVATIVES AS ADENOSIN ANTAGONISTS THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, U.S. DEPARTMENT OF COMMERCE (US) 1990-11-01 WO disclosed