SCHEMBL9258370

SCHEMBL9258370

COC(=O)COC(C)N1CCC(C(=O)c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 15/20 0.62
TACR1 P25103 2/20 0.62
TACR2 P21452 1/20 0.62
TP53 P04637 1/20 0.46
KCNH2 Q12809 1/20 0.46
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.44
CHRM1 P11229 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SSTR5 P35346 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9268866 0.85 HRH1 (0.43) HRH1TACR1TACR2ALDH1A1
SCHEMBL9258364 0.83 HRH1 (0.71) HRH1TACR1TACR2
SCHEMBL9260568 0.82 HRH1 (0.48) HRH1TACR1TACR2KCNH2CHRM1
SCHEMBL9260700 0.81 HRH1 (0.42) HRH1TACR1TACR2TP53ALDH1A1
SCHEMBL9264751 0.81 HRH1 (0.72) HRH1TACR1TACR2TP53KCNH2
SCHEMBL9259609 0.79 HRH1 (0.67) HRH1TACR1TACR2TP53KCNH2
SCHEMBL9282529 0.79 HRH1 (0.40) HRH1TACR1TACR2ALDH1A1LMNA
SCHEMBL9196229 0.78 HRH1 (0.66) HRH1TACR1TACR2TP53KCNH2
SCHEMBL9266568 0.78 HRH1 (0.66) HRH1TACR1TACR2TP53KCNH2
SCHEMBL9258366 0.78 HRH1 (0.63) HRH1TACR1TACR2TP53KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US claimed
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed