SCHEMBL9259308

SCHEMBL9259308

COC(=O)CSc1ccc(-c2nc(-c3ccc(C(=N)N)cc3)c[nH]2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TP53 P04637 1/20 0.36
GRK6 P43250 1/20 0.36
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
MAPT P10636 4/20 0.36
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
POLB P06746 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GAA P10253 2/20 0.35
CYP1A2 P05177 1/20 0.35
GLA P06280 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254922 0.87 GRK6 (0.42) GRK6ITGB3ITGA2BMAPTKDM4E
SCHEMBL9568559 0.82 F2 (0.41) ITGB3ITGA2B
SCHEMBL9253478 0.82 KLK1 (0.38) ITGB3ITGA2BNQO2
SCHEMBL9257084 0.82 F2 (0.41) ITGB3ITGA2B
Hydrochloric Acid SCHEMBL9254356 0.81 F2 (0.40) ITGB3ITGA2B
SCHEMBL9257715 0.81 NQO2 (0.35) ITGB3ITGA2BNQO2
SCHEMBL9254303 0.80 TMPRSS15 (0.43) SMN1; SMN2ITGB3ITGA2BPOLB
SCHEMBL9257749 0.80 PHGDH (0.37) ITGB3ITGA2BKDM4EALDH1A1GLA
SCHEMBL9568477 0.80 TMPRSS15 (0.38) ITGB3ITGA2BNQO2
SCHEMBL9256770 0.79 ITGB3 (0.35) ITGB3ITGA2BKDM4EALDH1A1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed