SCHEMBL9259459

SCHEMBL9259459

Clc1ccc(-c2nn(CCc3ncc[nH]3)c3ccncc23)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 6/20 0.38
MAPT P10636 1/20 0.35
TAAR1 Q96RJ0 2/20 0.34
CDC7 O00311 1/20 0.34
CDK2 P24941 1/20 0.34
CSNK2A2 P19784 1/20 0.33
CSNK2B P67870 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
PKM P14618 1/20 0.32
HPGD P15428 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TERT O14746 1/20 0.32
AOC3 Q16853 2/20 0.32
KCNH2 Q12809 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9255091 0.89 NAMPT (0.33) NAMPTTAAR1MAP4K4EGFRFRK
SCHEMBL9257063 0.88 HSD17B10 (0.40) TAAR1ALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL9302703 0.78 CSNK2A2 (0.39) NAMPTMAPTCDC7CDK2CSNK2A2
SCHEMBL8138744 0.77 CYP2D6 (0.42) NAMPTMAPTCDC7CDK2ALDH1A1
SCHEMBL9264217 0.77 NAMPT (0.36) NAMPTMAPTCDC7CDK2CSNK2A2
SCHEMBL8135725 0.76 LTA4H (0.39) NAMPTMAPTCDC7CDK2CSNK2A2
SCHEMBL8137068 0.75 CYP2D6 (0.49) NAMPTMAPTKDM4EKCNH2CYP1A2
SCHEMBL9305127 0.75 MERTK (0.41) NAMPTMAPTCDC7CDK2CSNK2A2
SCHEMBL8136501 0.75 MAPT (0.40) NAMPTMAPTCDC7CDK2CSNK2A2
SCHEMBL9259487 0.73 TP53 (0.44) ALDH1A1KDM4ENPC1KCNH2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed
US-5428169-A Antidepressants, treating compulsive disorders, stuttering, trichotillomania HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1995-06-27 US disclosed
US-5380847-A Reaction of 1-methylpiperidine-4-hydrazine, ketone and titanium isopropoxide to form hydrazone HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1995-01-10 US disclosed
EP-0594001-A1 Pyrazolo 4,3-c pyridines, a process for their preparation and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1994-04-27 EP disclosed
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US disclosed
US-5264576-A Antiserotonin agents, antidepressants and obsessive-compulsive disorders HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1993-11-23 US disclosed