SCHEMBL9259512

SCHEMBL9259512

O=C(O)c1sc2ccc(Cl)cc2c1CNCCC1CCN(Cc2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.50
BCHE P06276 4/20 0.50
CHRM4 P08173 7/20 0.49
MAOB P27338 3/20 0.48
MAOA P21397 2/20 0.48
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254634 0.90 MAOB (0.51) ACHEBCHECHRM4MAOBMAOA
SCHEMBL9261890 0.85 ACHE (0.51) ACHEBCHECHRM4MAOBMAOA
SCHEMBL9259505 0.76 KDM4E (0.51)
SCHEMBL9260014 0.74 CNR1 (0.56) ACHEBCHECHRM4MAOBMAOA
SCHEMBL7593860 0.70 ACHE (0.54) ACHEBCHE
SCHEMBL9260634 0.70 ACHE (0.54) ACHEBCHECHRM4MAOBMAOA
SCHEMBL9251113 0.70 ACHE (0.54) ACHEBCHECHRM4MAOBMAOA
SCHEMBL9251812 0.70 ACHE (0.64) ACHEBCHECHRM4MAOBMAOA
SCHEMBL220628 0.69 ACHE (0.58) ACHEBCHE
SCHEMBL4591300 0.69 DRD2 (0.52) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed