SCHEMBL9254634

SCHEMBL9254634

Cc1ccc2sc(C(=O)O)c(CNCCC3CCN(Cc4ccccc4)CC3)c2c1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.51
ACHE P22303 6/20 0.49
BCHE P06276 5/20 0.49
CHRM4 P08173 4/20 0.47
MAOA P21397 1/20 0.47
KCNH2 Q12809 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9261890 0.93 ACHE (0.51) MAOBACHEBCHECHRM4MAOA
SCHEMBL9259512 0.90 ACHE (0.50) MAOBACHEBCHECHRM4MAOA
SCHEMBL9251113 0.80 ACHE (0.54) MAOBACHEBCHECHRM4MAOA
SCHEMBL222020 0.79 ACHE (0.56) ACHEBCHE
SCHEMBL9260634 0.79 ACHE (0.54) MAOBACHEBCHECHRM4MAOA
SCHEMBL9254627 0.78 KDM4E (0.51) MAOBACHECHRM4
SCHEMBL9255566 0.75 ACHE (0.51) MAOBACHEBCHEMAOA
SCHEMBL4709902 0.75 DRD2 (0.51) MAOBACHEBCHE
SCHEMBL7593860 0.72 ACHE (0.54) ACHEBCHE
SCHEMBL9251812 0.71 ACHE (0.64) MAOBACHEBCHECHRM4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed