SCHEMBL9263103

SCHEMBL9263103

Nc1ccc(F)cc1-c1cc[nH]n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
CCNE2 O96020 2/20 0.39
CCNE1 P24864 2/20 0.39
CDK2 P24941 2/20 0.39
IDO1 P14902 3/20 0.36
KEAP1 Q14145 1/20 0.34
NPC1 O15118 3/20 0.34
NOS3 P29474 2/20 0.33
AXL P30530 1/20 0.33
GFER P55789 1/20 0.33
ALPL P05186 2/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PARP1 P09874 1/20 0.31
PARP10 Q53GL7 1/20 0.31
BACE1 P56817 1/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3846622 0.81 ALPL (0.35) ALDH1A1IDO1NPC1ALPLKDM4E
SCHEMBL27660921 0.79 IDO1 (0.38) IDO1NPC1ALPLPARP1PARP10
SCHEMBL100881 0.79 IDO1 (0.49) ALDH1A1IDO1NPC1MEN1USP2
SCHEMBL13963717 0.79 NISCH (0.45) CCNE1CDK2IDO1NPC1ALPL
SCHEMBL9038568 0.79 GPR35 (0.50) ALDH1A1IDO1KDM4EGAAHSD17B10
SCHEMBL14400038 0.79 IDO1 (0.58) ALDH1A1CDK2IDO1KDM4EHSD17B10
SCHEMBL988594 0.78 ALPL (0.48) IDO1NPC1ALPLCYP1A2CYP3A4
SCHEMBL30341309 0.76 FYN (0.34)
SCHEMBL7157001 0.76 CCNT1 (0.37) CDK2KEAP1ALPLPARP1
SCHEMBL22684363 0.75 ALOX5AP (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5387585-A Treating epilepsy, anxiety, sleep disorders, schizophrnia, senile dementia HOFFMANN-LA ROCHE INC. (US) 1995-02-07 US disclosed
EP-0519307-A2 Tetracyclic Imidazodiazepines F. HOFFMANN-LA ROCHE AG (CH) 1992-12-23 EP disclosed