SCHEMBL9260920

SCHEMBL9260920

O=C(O)Cn1c(C(=O)C2CCNCC2)nc2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
HSD17B10 Q99714 1/20 0.50
APEX1 P27695 1/20 0.49
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
PTGDR2 Q9Y5Y4 4/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7887857 0.86 HTR3A (0.52) KDM4E
SCHEMBL9695580 0.86 POLB (0.60) KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL9260978 0.85 KDM4E (0.50) KDM4EHSD17B10APEX1ALDH1A1HPGD
Bromide SCHEMBL3553550 0.85 POLB (0.59) KDM4EHSD17B10ALDH1A1HPGD
SCHEMBL7468259 0.83 HTR3A (0.54) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL7470479 0.81 HRH1 (0.50) KDM4EHSD17B10
SCHEMBL7474308 0.81 HRH1 (0.62)
SCHEMBL7469554 0.80 HRH1 (0.49) KDM4EHSD17B10ALDH1A1MEN1KMT2A
SCHEMBL7954906 0.80 HRH1 (0.52) KDM4EALDH1A1
SCHEMBL7465508 0.79 HRH1 (0.41) ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5389634-A Treating arterial hypertension, relaxing uterus, prevention of post-angioplastic restenosis ROUSSEL-UCLAF (FR) 1995-02-14 US disclosed
US-5380731-A Antiallergic compounds MERRELL DOW PHARMACEUTICALS INC. (US) 1995-01-10 US disclosed
EP-0561973-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-29 EP disclosed
WO-1992010491-A1 ANTIALLERGIC COMPOUNDS MERRELL DOW PHARMACEUTICALS INC. (US) 1992-06-25 WO disclosed