SCHEMBL9268779

SCHEMBL9268779

CN(C)C(=O)C(N)(C#N)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.45
DRD3 P35462 6/20 0.45
DRD4 P21917 4/20 0.45
DRD2 P14416 5/20 0.40
CYP2D6 P10635 3/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP3A4 P08684 2/20 0.38
ALDH1A1 P00352 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
KIF11 P52732 1/20 0.35
KCNN4 O15554 3/20 0.35
CYP2C19 P33261 2/20 0.35
MEN1 O00255 1/20 0.35
CYP2C9 P11712 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
HIF1A Q16665 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9268675 0.79 OPRM1 (0.47) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL10346433 0.75 OPRM1 (0.44) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL375036 0.70 OPRM1 (0.53) OPRM1DRD3DRD4DRD2MAPT
SCHEMBL6073343 0.70 OPRM1 (0.53) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL5642972 0.70 KMT2A (0.57) OPRM1DRD3DRD4DRD2CYP1A2
SCHEMBL10814384 0.70 OPRM1 (0.53) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL6073374 0.68 CYP1A2 (0.59) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL16158180 0.68 OPRM1 (0.51) OPRM1DRD3DRD4DRD2MAPT
SCHEMBL6309263 0.68 OPRM1 (0.65) OPRM1DRD3DRD4DRD2CYP2D6
SCHEMBL11005256 0.68 KMT2A (0.50) OPRM1DRD3DRD4DRD2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5436264-A Adrenergic blocking agents for vasoconstriction and hypotensive agents SYNTEX (U.S.A.) INC. (US) 1995-07-25 US disclosed