SCHEMBL9278686

SCHEMBL9278686

NC(=O)c1nocc1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 4/20 0.36
PTGS2 P35354 2/20 0.34
ALDH1A1 P00352 5/20 0.33
ADORA2A P29274 1/20 0.33
TBXA2R P21731 1/20 0.33
KDM4E B2RXH2 4/20 0.33
NPC1 O15118 2/20 0.33
PPARG P37231 1/20 0.33
NCOA2 Q15596 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RAB9A P51151 1/20 0.33
LDHA P00338 1/20 0.32
MAPT P10636 3/20 0.31
ALOX15 P16050 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
BLM P54132 1/20 0.31
AGER Q15109 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3039398 0.87 MAPT (0.33) IKBKBPTGS2ALDH1A1ADORA2AKDM4E
SCHEMBL8595148 0.85 ALDH1A1 (0.39) PTGS2ALDH1A1KDM4ENPC1LDHA
SCHEMBL9567818 0.79 PTGS2 (0.34) PTGS2ALDH1A1KDM4ENPC1LDHA
Valine SCHEMBL9429680 0.75 SLC7A5 (0.46) PTGS2
SCHEMBL163532 0.74
SCHEMBL17570173 0.74
SCHEMBL1790158 0.72
SCHEMBL29366578 0.72
SCHEMBL3348565 0.72
SCHEMBL161729 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1051074-C Isoxazole-4-carboxamides and hydroxyalkylidenecyanoacetamides pharmaceuticals containing these compounds and their use HOECHST AG (DE) 2000-04-05 CN disclosed
US-5378680-A Dicarboximides and their use as herbicides BASF AKTIENGESELLSCHAFT (DE) 1995-01-03 US disclosed
US-5276160-A Amidation of primary or secondary amines BASF AKTIENGESELLSCHAFT (DE) 1994-01-04 US disclosed
US-5264580-A Reaction of hydroximyl chlorides and beta-keto acids or esters, cyclization BASF AKTIENGESELLSCHAFT (DE) 1993-11-23 US disclosed
US-5176739-A Plant growth regulators BASF AKTIENGESELLSCHAFT (DE) 1993-01-05 US disclosed
CN-1056684-A Different  azoles-4-carboxylic acid amides and hydroxy alkylidene Malonamide nitrile contains the medicine of these compounds and their application HOECHST AG (DE) 1991-12-04 CN disclosed